[ACS] Lead Optimizationof Multimutant KRAS Switch-II PocketMacrocyclic Inhibitors via Isosteric Replacement to Improve ADME andOral Exposure

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xiehb88 发表于 2026-9-4 17:11:03 | 显示全部楼层 |阅读模式
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期刊:Journal of Medicinal Chemistry

文献作者:Dean P. Phillips; Phil B. Alper; Dmitry Borkin; Dong Han; Sarah E. Kochanek; Jitendra Gurjar; Casey J. N. Mathison; John M. Nelson; Wei Pei; Bao Ngoc Nguyen; Timothy Hoffman; Barun Okram; Truc N. Nguyen; Songchun Jiang; Brian T. Masick; Zhicheng Wang; Charles Y. Cho; Hong Yin; Yu Chen; Jose Juarez; Yong Jia; Vicki Zhou; Guoxun Liu; Clifford Wright; Trish Nguyen; Deborah A. Knee; Qian Liu; Jun Liu; Jie Li; Cyrus Virata; Cesar de Oliveira; Michael DiDonato; Badry Bursulaya; Agnes Vidal-Biggart; David H. Jones; Darbi Witmer; Carolyn Chu; Hong Jin; Ananda Herath; Wendy Richmond; Todd Groessl; Michael Shapiro; Kathleen Effenberger; Konrad Arroyo; Angela Bretz; Ayako Honda; William P. Gordon; Valentina Molteni; Jacob R. Haling

出版日期:--

DOI号:10.1021/acs.jmedchem.6c01454

下载链接:https://pubs.acs.org/jmcmar/arti ... medchem.6c01454.pdf

文献链接:https://doi.org/10.1021/acs.jmedchem.6c01454

当前文献来源于 American Chemical Society (ACS)。


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